DMARDs

red flags in bloods

indicates urgent referral to rheum from primary care

Main risks:

  • agranulocytosis
  • impaired renal function
  • impaired liver function

FBC

  • White cell count lower than 3.5 x 109/L.
  • Mean cell volume higher than 105 fL. 
    • Check B12, folate, and thyroid-stimulating hormone levels.
    • If abnormal, treat; if normal, discuss with specialist team.
  • Neutrophils lower than 1.6 x 109/L.
  • Unexplained eosinophilia higher than 0.5 x 109/L
  • Platelet count lower than 140 x 109/L.

U+E

  • Creatinine has increased by more than 30% over 12 months and/or calculated glomerular filtration rate (GFR) is lower than 60 mL/min.
    • Repeat in 1 week.
    • If still more than 30% from baseline, withhold and discuss with specialist team.

Liver function tests

  • Alanine aminotransferase (ALT) and/or aspartate transaminase (AST) higher than 100 U/L.
  • Unexplained reduction in albumin lower than 30 g/L.

Others

  • Blood pressure higher than 140/90mmHg. 
    • If on cislosporin, stop treatment and discuss with specialist team. 
    • If on other DMARDs, manage in accordance with hypertension guidelines. 
  • Urinary protein 2+ or more.
    • Check mid-stream urine sample.
    • If evidence of an infection, treat appropriately; if sterile and 2+ proteinuria or more persists on two consecutive measurements, withhold until discussed with specialist team.

routine monitoring

azathioprine, mycophenolate, sulfasalazine

Monitoring Frequency
FBC - Every 2 weeks until dose is stable for 6 weeks, then monthly for 3 months.
- Thereafter, at least every 12 weeks.
- Monitor more frequently in people at higher risk of toxicity.
- If dose is increased, monitor every 2 weeks until dose is stable for 6 weeks, then revert to previous schedule.
Renal function: creatinine/calculated GFR
LFTs: ALT and/or AST and albumin

ciclosporin, tacrolimus, leflunomide

Monitoring Frequency
FBC - Every 2 weeks until dose is stable for 6 weeks, then monthly.
- People who have been stable for 12 months can be considered for reduced monitoring frequency (every 3 months) on an individual basis.
- Monitor more frequently in people at higher risk of toxicity.
- If the dose is increased, monitor every 2 weeks until dose is stable for 6 weeks, then revert to previous schedule.
Renal function: creatinine/calculated GFR
LFTs: ALT and/or AST and albumin
Blood glucose
Blood pressure

Leflunomide - include weight

cyclophosphamide, penicillamine

Monitoring Frequency
FBC - 10 days after each pulse therapy.
- Blood tests repeated immediately prior to the next pulse.
LFTs: ALT and/or AST and albumin
Urinalysis

Penicillamine - include renal function

hydroxychloroquine

Monitoring Frequency
Renal function - Annually in people aged over 70 years old and in those with pre-existing renal impairment, hypertension, and/or diabetes.
Eye assessment (ideally including optical coherence tomography) - Annually for all people who have taken hydroxychloroquine for greater than 5 years.
- Annual monitoring may be commenced before 5 years of treatment if additional risk factors for retinal toxicity exist, such as:
- Concomitant tamoxifen therapy, impaired renal function (estimated glomerular filtration rate less than 60 mL/minute/1.73 m2) or
- High-dose therapy (greater than 5 mg/kg/day of hydroxychloroquine).

advice

  • ↑ susceptibility to infection in 1st 6/12